BET Inhibitors

BET Inhibitors


Bromodomain and Extra-Terminal motif (BET) inhibitors are a class of small molecule drugs that reversibly bind the bromodomains of BET proteins BRD2, BRD3, BRD4, and BRDT. These BET inhibitors prevent protein-protein interaction between BET proteins and acetylated histones and transcription factors. Dysregulated bromodomains of BET proteins are frequently found in cancer showing aberrant chromatin remodeling and gene expression.

Catalog Product Name Structure M.W. Purity Pricing
BET Inhibitors
BP-21590(+)JQ-1Molecular structure of the compound: (+)JQ-1457.0Pricing
BP-40229(+)-JQ1 carboxylic acidMolecular structure of the compound: (+)-JQ1 carboxylic acid400.998%Pricing
BP-23442I-BET 762Molecular structure of the compound: I-BET 762423.998%Pricing
BP-23376MS-436Molecular structure of the compound: MS-436383.498%Pricing
BP-23384BI-2536Molecular structure of the compound: BI-2536521.795%Pricing
BP-23380RVX-208Molecular structure of the compound: RVX-208370.498%Pricing
BP-25347BAY 299Molecular structure of the compound: BAY 299429.5Pricing
BP-25348BAZ2-ICRMolecular structure of the compound: BAZ2-ICR357.4Pricing
BP-25349BI 9564Molecular structure of the compound: BI 9564353.4Pricing
BP-25350BromosporineMolecular structure of the compound: Bromosporine404.5Pricing
BP-25351CPI 203Molecular structure of the compound: CPI 203399.9Pricing
BP-25352GSK 2801Molecular structure of the compound: GSK 2801371.5Pricing
BP-25353GSK 5959Molecular structure of the compound: GSK 5959394.5Pricing
BP-25354GSK 6853Molecular structure of the compound: GSK 6853409.5Pricing
BP-25356I-BRD9Molecular structure of the compound: I-BRD9497.6Pricing
BP-25365NI 57Molecular structure of the compound: NI 57383.4Pricing
BP-25368OTX 015Molecular structure of the compound: OTX 015492.0Pricing
BP-25371PFI 1Molecular structure of the compound: PFI 1347.4Pricing
BP-25372PFI 3Molecular structure of the compound: PFI 3321.4Pricing
BP-25373PFI 4Molecular structure of the compound: PFI 4380.5Pricing
BP-25374SGC-CBP30Molecular structure of the compound: SGC-CBP30509.1Pricing
BP-25377XMD 8-92Molecular structure of the compound: XMD 8-92474.6Pricing
BP-27845N-[3-Chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amineMolecular structure of the compound: N-[3-Chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amine505.7Pricing
BP-27851dBET1Molecular structure of the compound: dBET1785.3Pricing
BP-27856l-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-lHpyrazolo [3,4-d]pyrimidin-l-yl]-l-piperidinyl]-2-propyn-l-oneMolecular structure of the compound: l-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-lHpyrazolo [3,4-d]pyrimidin-l-yl]-l-piperidinyl]-2-propyn-l-one438.5Pricing
BP-278574-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)quinazolin-6-yl)phenolMolecular structure of the compound: 4-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)quinazolin-6-yl)phenol471.9Pricing